Letrozole

Letrozole for sale in USA

Letrozole is an antitumor agent in the group of non-steroidal aromatase inhibitors (inhibitor of estrogen synthesis). It is known that many steroid drugs aromatize into estrogens, therefore, there is a risk of men who take steroids developing hormones that act in a female fashion causing gynecomastia, fluid accumulation and fat deposition. In such cases, it is necessary to use an antiestrogen that prevents and blocks the development of such consequences. Through selective aromatase inhibition, Letrozole is able to block estrogen biosynthesis in peripheral and tumor tissues. The drug inhibits aromatase by simultaneous binding to cytochrome P450 iron with reduced estrogen synthesis in tissues.

The Effectiveness of the drug: Advantages of buying Letrozole for your cycle

Bodybuilders and athletes who take anabolic steroids will generally favor the use of Letrozole because of the drug’s exceptional capabilities:

• Letrozole has the ability to eliminate rising estrogen levels at the root cause (the aromatization process).
• It is an inhibitor of high selectivity (superior to Fadrozole, Anastrozole, etc.) compared to aromatase.
• Letrozole is rapidly and almost completely absorbed from the gastrointestinal tract, its bioavailability is 99.9%.
• It is promptly and widely distributed in tissues.
• The drug does not cause disruption of steroidogenesis in the adrenal glands and androstenedione level in plasma.
• Letrozole may be administered independently of meals.
• The pharmacokinetics of Letrozole is independent of age.

The use of Letrozole

The standard dose for Letrozole tablets is 1.25-2.5mg daily. Even a dose as small as this is effective enough to reduce the circulating estrogen levels by around 98%. The dosage can be adjusted to suit each user’s tolerance, each individual should slowly adjust their dose depending on how they feel and how their body is responding to the drug. Even 1.25mg daily is an overly high dose for some anabolic steroid users, so in this case, considering the half-life of Letrozole is 2-4 days, the frequency of use can be reduced from every day to every 2-3 days if needed.